托烷司瓊
Product Name: Tropisetron
CAS號:89565-68-4
分子式:C17H20N2O2
分子量:284.35
貯存: 儲存溫度-20°C
可溶性: DMSO
生化和生理學(xué)機(jī)理:
Tropisetron is a selective 5-HT3 receptor antagonist and α7-nicotinic receptor agonist with an IC50 of 70.1 ± 0.9 nM for 5-HT3 receptor. It is used mainly as an antiemetic to treat nausea and vomiting following chemotherapy, although it has been used experimentally as an analgesic in cases of fibromyalgia.